A one-pot radioiodination of aryl amines via stable diazonium salts: preparation of 125I-imaging agents
نویسندگان
چکیده
منابع مشابه
A one-pot radioiodination of aryl amines via stable diazonium salts: preparation of 125I-imaging agents.
An operationally simple, one-pot, two-step tandem procedure that allows the incorporation of radioactive iodine into aryl amines via stable diazonium salts is described. The mild conditions are tolerant of various functional groups and substitution patterns, allowing late-stage, rapid access to a wide range of 125I-labelled aryl compounds and SPECT radiotracers.
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ژورنال
عنوان ژورنال: Chemical Communications
سال: 2017
ISSN: 1359-7345,1364-548X
DOI: 10.1039/c7cc06211g